- Process research for multikilogram production of etamicastat: A novel dopamine β-hydroxylase inhibitor
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In order to develop a manufacturing route to etamicastat, three synthetic approaches to the pivotal chiral 3-aminochroman intermediate have been studied as well as four methods for the construction of the 2-aminoethyl imidazolethione fragment. The evoluti
- Beliaev, Alexandre,Wahnon, Jorge,Russo, Domenico
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p. 704 - 709
(2012/07/03)
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- PROCESS
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Compounds of formula I, V, VI and II, and processes for their preparation, wherein R1, R2 and R3 are the same or different and signify hydrogens, halogens, alkyl, alkyloxy, hydroxy, nitro, alkylcarbonylamino, alkylamino or
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Page/Page column 29
(2009/06/27)
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