Synthesis, Absolute Configuration and Local Anaesthetic Activity of the Enantiomers of α- and β-Methylprocaine
Optically active forms of 1-(diethylaminomethyl)ethyl 4-aminobenzoate (α-methylprocaine) (1) and 2-(diethylamino)propyl 4-aminobenzoate (β-methylprocaine) (2) of known absolute configuration have been prepared.The enantiomers show no stereoselectivity in
Bell, Kevin H.,Fullick, Graeme
p. 1429 - 1433
(2007/10/02)
Regiospecific Conversion of Oxiranes into Primary Alcohols via Reaction with Organotin Derivatives