1159685-85-4Relevant articles and documents
8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones: Dual-acting 5-HT1 receptor antagonists and serotonin reuptake inhibitors-Part II
Bromidge, Steven M.,Bertani, Barbara,Borriello, Manuela,Bozzoli, Andrea,Faedo, Stefania,Gianotti, Massimo,Gordon, Laurie J.,Hill, Matthew,Zucchelli, Valeria,Watson, Jeannette M.,Zonzini, Laura
supporting information; experimental part, p. 2338 - 2342 (2009/12/31)
8-[2-(4-Aryl-1-piperazinyl)ethyl]-2H-1,4-benzoxazin-3(4H)-ones have been identified as highly potent 5-HT1A/B/D receptor antagonists with and without additional SerT activity and a high degree of selectivity over hERG potassium channels. Modula
