1416767-44-6Relevant articles and documents
Substrate scope in the direct imine acylation of ortho-substituted benzoic acid derivatives: The total synthesis (±)-cavidine Dedicated to the memory of Sandy McKillop - Colleague, mentor, collaborator and friend
Kitsiou, Christiana,Unsworth, William P.,Coulthard, Graeme,Taylor, Richard J.K.
, p. 7172 - 7180 (2015/06/23)
The direct imine acylation (DIA) and subsequent cyclisation of a range of imines with ortho-substituted benzoic acid derivatives is described. Variation in the coupling reagents, imine and benzoic acid were all examined. The DIA procedure was also applied in the total synthesis of (±)-cavidine.