28944-98-1Relevant articles and documents
Metal-free direct amidation of peptidyl thiol esters with α-amino acid esters
Chen, Hao,He, Maomao,Wang, Yaya,Zhai, Linhui,Cui, Yongbo,Li, Yangyan,Lee, Yan,Zhou, Haibing,Hong, Xuechuan,Deng, Zixin
, p. 2723 - 2726 (2011/11/06)
Metal-free direct amidation of peptidyl thiol esters with α-amino acid esters in the presence of bis(trimethylsilyl) acetamide (BSA) has been developed. This general method provides convenient access to N-protected peptides in good yields under mild condi
Dehydrogenation of Indolines to Indoles via Azasulphonium Salts or N-Chloramines
Kawase, Masami,Miyake, Yuko,Kikugawa, Yasuo
, p. 1401 - 1404 (2007/10/02)
The dehydrogenation of indolines to indoles without using mineral oxidising reagents is described.The conversion was achieved via either azasulphonium salts or N-chloramines, the former route involving milder conditions but a more complex procedure.