LY 2183240 Price
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1. LY 2183240 HPLC
LY 2183240 HPLC is a potent inhibitor of anandamide uptake which inhibits FAAH (IC50=2.1 nM) and some other brain serine proteases. LY 2183240 HPLC elevates brain anandamide levels and shows efficacy in a rodent model of persistent pain (ED50=1.37 mg/kg). Regioisomer 2-5 of LY2183240 is less active. LY 2183240 HPLC is more potent than N-(4-Hydroxyphenyl)-arachidonylamide (AM-404), which inhibits anandamide transport at IC50=1mM.
2. Biological activity of LY 2183240 HPLC
Novel and highly potent blocker of anandamide uptake (IC50 = 270 pM). Inhibits fatty acid amide hydrolase (FAAH) activity (IC50 = 12.4 nM). Following i.p. administration in rats, increases brain anandamide concentration and exerts antinociceptive effects in formalin model of pain.
3. LY 2183240 Price
LY 2183240 is also called 5-(4-Biphenylylmethyl)-N,N-dimethyl-1H-tetrazole-1-carboxamide, MN-25. At present, LY 2183240 price is stable. The statistic offered by Shanghai Tangfang Biotechnology Co., Ltd is for reference: $209 (10 mg). If you want to get the latest LY 2183240 price, please contact with the manufacture.
Verified Supplier
Shanghai Tangfang Biotechnology Co., Ltd.
- Country: China (Mainland)
- Year Established: 2010
- Business type: Manufacturers
- Integral:
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