- Mosquito acetylcholinesterase as a target for novel phenyl-substituted carbamates
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New insecticides are needed for control of disease-vectoring mosquitoes and this research evaluates the activity of new carbamate acetylcholinesterase (AChE) inhibitors. Biochemical and toxicological characterization of carbamates based on the parent stru
- Mutunga, James M.,Ma, Ming,Chen, Qiao-Hong,Hartsel, Joshua A.,Wong, Dawn M.,Ding, Sha,Totrov, Max,Carlier, Paul R.,Bloomquist, Jeffrey R.
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- Tetrazolinone compound, and use therefor
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A tetrazolinone compound represented by formula (1) (in the formula, R1, R2, R3, and R11 each represent a halogen atom, a C1-C6 alkyl group, or the like; R4 and R5 each represent a hydrogen atom, a halogen atom, a C1-C3 alkyl group, or the like; R6 represents a C1-C3 alkyl group which may have one or more halogen atoms, or the like; R7 R8, and R9 each represent a hydrogen atom, a halogen atom, or the like; R10 represents a C1-C3 alkyl group, or the like; and R12 represents a phenyl group which may have one or more atoms or groups selected from group (P3), a phenoxy group which may have one or more atoms or groups selected from group (P3), or the like). The tetrazolinone compound has an excellent pest-control effect.
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Paragraph 1355; 1356; 1357; 1358
(2016/10/08)
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- TETRAZOLINONE COMPOUND AND USE THEREOF
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A tetrazolinone compound represented by formula (1): Wherein R1, R2, R3, and R11 each represents a halogen atom, a C1-C6 alkyl group, etc.; R4 and R5 each represents a hydrogen atom, a halogen atom, a C1-C3 alkyl group, etc.; R6 represents a C1-C3 alkyl group optionally having one or more halogen atoms, etc.; R7, R8, and R9 each represents a hydrogen atom, a halogen atom, etc.; R10 represents a C1-C3 alkyl group, etc.; and R12 represents a phenyl group optionally having one or more atoms or groups selected from Group P3, a phenoxy group optionally having one or more atoms or groups Group P3, etc., has excellent control activity against pests.
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Paragraph 0709; 0710
(2016/07/05)
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- An efficient synthetic route to novel 3-alkyl- and 3-aryl-4-iodophenols
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An efficient method for the preparation of novel 3-alkyl-and 3-aryl-4-iodophenols from 3-alkyl- and 3-arylphenols is described. Georg Thieme Verlag Stuttgart.
- Hermann, Gesine J.,Annis, Michael C.,Edwards, Peter D.,Corrales, Marta,Diaz, Lucia,Goodnow, Robert A.
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p. 221 - 224
(2008/12/20)
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- Compounds having activity as inhibitors of cytochrome P450RAI
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Compounds having Formula 2 wherein the symbols have the meaning defined in the specification are inhibitors of the cytochrome P450RAI (retinoic acid inducible) enzyme, and are used for treating diseases responsive to treatment by retinoids.
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Page column 108
(2010/01/31)
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- Compounds having activity as inhibitors of cytochrome P450RAI
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Compounds having Formula 8 wherein the symbols have the meaning defined in the specification are inhibitors of the cytochrome P450RAI (retinoic acid inducible) enzyme, and are used for treating diseases responsive to treatment by retinoids.
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Page column 40, 109
(2010/11/29)
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- Compounds having activity as inhibitors of cytochrome P450RAI
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Compounds having Formula 1 wherein the symbols have the meaning defined in the specification are inhibitors of the cytochrome P450RAI (retinoic acid inducible) enzyme, and are used for treating diseases responsive to treatment by retinoids.
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Page column 110
(2010/01/31)
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- Preparation of 4-Bromo- and 4-Chloro-3-t-butylphenol
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4-Bromo- and 4-Chloro-3-butylphenol, two potent fungistatics, were prepared in an efficient 3-step synthesis from commercially available materials.Crucial to the synthesis is the use of halo-substituents as positional protective groups.
- Fukata, Gouki,Kubota, Yukihiro,Mataka, Shuntaro,Thiemann, Thies,Tashiro, Masashi
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p. 592 - 594
(2007/10/02)
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- Tert-Butyl-halophenols
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3-tert-Butyl-4-halophenols which are useful as intermediates for preparing compounds having medical or agricultural activities.
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