Bioorganic and Medicinal Chemistry Letters p. 3156 - 3161 (2006)
Update date:2022-08-02
Topics:
Penning, Thomas D.
Khilevich, Albert
Chen, Barbara B.
Russell, Mark A.
Boys, Mark L.
Wang, Yaping
Duffin, Tiffany
Engleman, V. Wayne
Finn, Mary Beth
Freeman, Sandra K.
Hanneke, Melanie L.
Keene, Jeffery L.
Klover, Jon A.
Nickols, G. Allen
Nickols, Maureen A.
Rader, Randall K.
Settle, Steven L.
Shannon, Kristen E.
Steininger, Christina N.
Westlin, Marisa M.
Westlin, William F.
We describe a series of pyrazole and isoxazole analogs as antagonists of the αvβ3 receptor. Compounds showed low to sub-nanomolar potency against αvβ3, as well as good selectivity against αIIbβ3<
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