21816-82-0Relevant articles and documents
Anti-infective and herbicidal activity of N-substituted 2-aminobenzothiazoles
Fajkusova, Dagmar,Pesko, Matus,Keltosova, Stanislava,Guo, Jiahui,Oktabec, Zbynek,Vejsova, Marcela,Kollar, Peter,Coffey, Aidan,Csollei, Jozef,Kralova, Katarina,Jampilek, Josef
, p. 7059 - 7068 (2012)
In this study, a series of N-substituted 2-aminobenzothiazoles was prepared according to a recently developed method. Twelve compounds were tested for their activity related to the inhibition of photosynthetic electron transport (PET) in spinach (Spinacia
An aerobic oxidative coupling approach for the synthesis of N-substituted 2-aminobenzothiazole derivatives using iron catalyst
Kumar, N. V. Anil,Kamath, Shailesha,Gaonkar, Santosh L.,Shetty, Nitinkumar S.
, p. 1697 - 1702 (2016)
A facile and convenient method was developed for the formation of novel N substituted 2-aminobenzothiazoles via an iron-catalysed condensation of 2-aminobenzothizole with different amines. This method is applicable for a wide range of aliphatic, aromatic and heterocyclic amines furnishing moderate yields of the corresponding products and thus rendering the methodology as a highly eco-friendly, inexpensive alternative to the existing methods.
Iron-Catalyzed Oxidative Amination of Benzylic C(sp3)–H Bonds with Anilines
Song, Yan-Ling,Li, Bei,Xie, Zhen-Biao,Wang, Dan,Sun, Hong-Mei
, p. 17975 - 17985 (2021/12/13)
Iron-catalyzed oxidative amination of benzylic C(sp3)–H bonds with anilines bearing electron-withdrawing groups (EWGs) or electron-donating groups (EDGs) is realized based on simple variations of N-substituents on imidazolium cations in novel ionic Fe(III) complexes. The structural modification of the imidazolium cation resulted in regulation of the redox potential and the catalytic performance of the iron metal center. Using DTBP as oxidant, [HItBu][FeBr4] showed the highest catalytic activity for anilines bearing EWGs, while [HIPym][FeBr4] was more efficient for EDG-substituted anilines. This work provides alternative access to benzylamines with the advantages of both a wide substrate scope and iron catalysis.
BENZOTHIAZOLE COMPOUNDS AND USES THEREOF
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Page/Page column 69, (2021/12/29)
The present invention features compounds useful in the treatment of neurological disorders. The compounds of the invention, alone or in combination with other pharmaceutically active agents, can be used for treating or preventing neurological disorders.