1243565-51-6Relevant articles and documents
2-And 3-phenylsulfonylindoles-synthetic equivalents of unsubstituted indole in n-alkylation reactions
Karchava,Shuleva,Ovcharenko,Yurovskaya
, p. 291 - 301 (2011/04/22)
The N-alkylation of 2- and 3-phenylsulfonylindoles under various conditions and the subsequent removal of the activating phenylsulfonyl group by reductive desulfonylation using Raney nickel leads to N-alkylindoles in high yield. 2-Phenylsulfonylindole readily undergoes the Mitsunobu reaction, while isomeric 3-phenylsulfonylindole is relatively inert under these conditions.
