179188-06-8Relevant articles and documents
Structure-Activity Relationships of the Peptide Kappa Opioid Receptor Antagonist Zyklophin
Joshi, Anand A.,Murray, Thomas F.,Aldrich, Jane V.
, p. 8783 - 8795 (2015)
The dynorphin (Dyn) A analogue zyklophin ([N-benzyl-Tyr1-cyclo(d-Asp5,Dap8)]dynorphin A(1-11)NH2) is a kappa opioid receptor (KOR)-selective antagonist in vitro, is active in vivo, and antagonizes KOR in the CNS
DTPA derivatives substituted in a novel way, their metal complexes, and their use in diagnosis and therapy
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, (2008/06/13)
The invention relates to new diethylenetriaminepentaacetic acid derivatives, their complexes and complex salts, that contain an element of atomic numbers 20-32, 39-51 or 57-83, pharmaceutical agents that contain these compounds and their use as contrast m
N-terminal alkylated derivatives of [D-Pro10]dynorphin A-(1-11) are highly selective for κ-opioid receptors [2]
Choi,Murray,DeLander,Caldwell,Aldrich
, p. 4638 - 4639 (2007/10/02)
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