2859-30-5Relevant articles and documents
Azide-Triggered Bicyclization of o-Alkynylisocyanobenzenes: Synthesis of Tetrazolo[1,5-a]quinolines
Khaikate, Onnicha,Soorukram, Darunee,Leowanawat, Pawaret,Pohmakotr, Manat,Reutrakul, Vichai,Kuhakarn, Chutima
, p. 7050 - 7057 (2019/11/11)
An efficient and rapid synthetic approach for the synthesis of tetrazolo[1,5-a]quinolines has been developed employing the reaction of o-alkynylisocyanobenzenes with sodium azide. The present strategy involved nucleophilic addition of azide to isocyanide followed by 6-endo cyclization. The reaction gives access to a collection of tetrazolo[1,5-a]quinolines with broad functional group in moderate to high yields under metal-, and base-free conditions.
Synthesis of quinolinones with palladium-catalyzed oxidative annulation between acrylamides and arynes
Wang, Weiguo,Peng, Xianglong,Qin, Xiaoyu,Zhao, Xiangyun,Ma, Chen,Tung, Chen-Ho,Xu, Zhenghu
, p. 2835 - 2841 (2015/03/18)
An unprecedented palladium-catalyzed oxidative annulation of acrylamides with benzyne precursors has been successfully developed. By using this mild "N-H activation/Heck reaction" method, a wide variety of quinolinones were conveniently prepared in one st
Synthesis of 4-Aryl-2-aminopyridine derivatives and related compounds
Pavlovic, Vladimir,Petkovic, Milos,Popovic, Stanimir,Savic, Vladimir
experimental part, p. 4249 - 4263 (2010/01/15)
A short, efficient, and high-yielding synthesis of 4-aryl-2-aminopyridine derivatives has been developed. The route employs two palladium-catalyzed processes, the Suzuki reaction and the Buchwald-Hartwig amination, as the key steps. The same approach has