750585-94-5Relevant articles and documents
INHIBITORS OF INDOLEAMINE 2,3-DIOXYGENASE
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Page/Page column 30; 31; 32, (2017/01/23)
Provided are compounds of formula (I) and pharmaceutically acceptable salts thereof, their pharmaceutical compositions, their methods of preparation, and methods for their use in the prevention and/or treatment of HIV; including the prevention of the prog
Psoromic acid is a selective and covalent rab-prenylation inhibitor targeting autoinhibited rabggtase
Deraeve, Celine,Guo, Zhong,Bon, Robin S.,Blankenfeldt, Wulf,DiLucrezia, Raffaella,Wolf, Alexander,Menninger, Sascha,Stigter, E. Anouk,Wetzel, Stefan,Choidas, Axel,Alexandrov, Kirill,Waldmann, Herbert,Goody, Roger S.,Wu, Yao-Wen
supporting information; experimental part, p. 7384 - 7391 (2012/06/30)
Post-translational attachment of geranylgeranyl isoprenoids to Rab GTPases, the key organizers of intracellular vesicular transport, is essential for their function. Rab geranylgeranyl transferase (RabGGTase) is responsible for prenylation of Rab proteins
Synthesis and structure-activity relationships of novel benzoxaboroles as a new class of antimalarial agents
Zhang, Yong-Kang,Plattner, Jacob J.,Freund, Yvonne R.,Easom, Eric E.,Zhou, Yasheen,Gut, Jiri,Rosenthal, Philip J.,Waterson, David,Gamo, Francisco-Javier,Angulo-Barturen, Inigo,Ge, Min,Li, Zhiya,Li, Lingchao,Jian, Yong,Cui, Han,Wang, Hailong,Yang, Jian
, p. 644 - 651 (2011/03/18)
A series of boron-containing benzoxaborole compounds was designed and synthesized for a structure-activity relationship investigation surrounding 7-(HOOCCH2CH2)-1,3-dihydro-1-hydroxy-2,1-benzoxaborole (1) with the goal of discovering